peptide wiki

GHRP-2

aka Growth Hormone Releasing Peptide-2

Growth Hormone Secretagogues

Mechanism

GHRP-2 (pralmorelin) is a synthetic hexapeptide ghrelin receptor agonist that stimulates pituitary growth hormone release. It is approved in Japan (Kaken Pharmaceutical, 2004) as a single-dose diagnostic agent for GH deficiency, but is NOT FDA-approved in the US and is research-only. Unlike ipamorelin, GHRP-2 is non-selective and modestly raises ACTH, cortisol, and prolactin.

Identification

CAS number158861-67-7
Molecular formulaC45H55N9O6
SequenceAAWFK
Typical dose100–300 mcg per injection, 2–3x daily, subcutaneous
Half-life~15–30 minutes

Vendors selling GHRP-2

VendorSizePriceListed purityTrust
Moglabs 5 mg $16.00 96
Ion Peptide 5 mg $29.00 95
Peptide Tech $18.99 94
Peptidology 10 mg $42.99 89
Qihang Peptide 87
Simple Peptide $39.00 85
Peptidegurus 5 mg 84
Peptidegurus 10 mg 84
Crystal Peptides 5 mg $24.96 66
Certified Peptides 10 mg $46.00 62
Peptiatlas 51
DongCheng Peptide 46
Mandy 5 mg $21.00 43
HongDa Peptide $29.00 43
HongDa Peptide $29.00 43
zztai Peptide Ltd 43
MJT peptides 5 mg $24.00 39
Alpha Omega $39.00
Atomik Labz 10 mg $39.00
Biotech Peptides 5 mg $20.00
Biotech Peptides 10 mg $39.00
Core Peptides 10 mg $20.00
Core Peptides 5 mg $20.00
Genetic Peptide 10 mg $40.00
Kimera Chems $21.99
Modern Research Peptides 10 mg $29.99
Oasis Labs 10 mg $47.00
Solution Peptides 10 mg $39.00
Solution Peptides 5 mg $19.00
Soma Peptides 10 mg $44.00

Research

Differential reversibility of anterior and posterior pituitary dysfunction in delayed recurrent pediatric Rathke's cleft cyst
Ogasawara A, Yamada S, Matsuoka G. · Endocrinology, diabetes & metabolism case reports (2026) · case-report

Summary Rathke's cleft cyst (RCC) is a benign sellar or suprasellar lesion increasingly detected by magnetic resonance imaging (MRI).

source →
Growth Hormone-Releasing Peptides: Investigation of Their Secondary Structure, Thermal Stability, and Model Membrane Interactions
Králík F, Kvíčalová A, Salaďáková A, Kuchař M, Setnička V. · Chirality (2026) ·

Growth hormone-releasing peptides (GHRPs) comprise a group of small synthetic peptides that can effectively influence growth hormone secretion both in humans and animals.

source →
Pituitary dysfunction in trans-sellar encephalocele: a two-case report and a literature review
Amano K, Seki Y, Koizumi S, Kawauchi Y, Yamashita M, Kurozumi K, Ichihara A, Kawamata T. · Endocrine journal (2026) · review

Trans-sellar encephalocele (TSE) is a rare congenital anomaly of the cranial base characterized by herniation of intracranial contents through the sellar floor. Although clinical presentations are diverse, the prevalence and characteristics of endocrine dysfunction due to hypothalamic-pituitary involvement are unclear.

source →
The emerging landscape of performance-enhancing peptides modulating GH-IGF1 axis: bridging the gap between clinical evidence and patient self-administration
Dominikowski A, Rękoś Z, Olejarz M, Szczepanek-Parulska E, Domin R, RuchaŁa M. · Frontiers in endocrinology (2026) · review

Performance-enhancing drugs (PEDs) marketed as "research compounds" include unregulated peptides intended to modulate the growth hormone-insulin-like growth factor-1 (GH-IGF-1) axis.

source →
Endocrine disorders in pediatric medulloblastoma survivors treated with X-ray or proton beam therapy: a single-institution retrospective study
Kaneko N, Morikawa S, Endo M, Hishimura N, Zhitong L, Yamaguchi T, Segoe H, Abe J, Oura K, Sawai S, Sugiyama M, Terashita Y, Hirabayashi S, Cho Y, Nakamura A, Ishi Y, Takao S, Mats, et al. · Endocrine journal (2026) · cohort

Medulloblastoma, a common pediatric central nervous system disease, is managed with surgery, chemotherapy, and craniospinal irradiation (CSI) delivered with either X-rays or protons. Proton-beam CSI, introduced to protect the surrounding tissues, may reduce endocrine toxicity.

source →
Behavioral Therapy Ameliorates Severe Obesity With Low Levels of Plasma GH and IGF-1: A Case Report
Yoshimichi G. · Clinical case reports (2026) ·

We encountered a patient with a body mass index of 50.7 kg/m 2 . Behavioral therapy was effective for preventing progression of health disturbance in this case. When coping with severe obesity, we must promote various tests to differentiate secondary obesity.

source →
On the road of dried blood spot sampling for antidoping tests: Detection of GHRP-2 abuse
Reverter-Branchat G, Segura J, Pozo OJ. · Drug testing and analysis (2021) ·

Dried blood spots (DBSs) sampling is gaining support by the antidoping community because of simplicity and cost-effective characteristics, especially in collection, transport, and storage. Nevertheless, DBS applicability demands specific studies for each of the analytes proposed for testing.

source →
Identification of a novel growth hormone releasing peptide (a glycine analogue of GHRP-2) in a seized injection vial
Popławska M, Błażewicz A. · Drug testing and analysis (2019) ·

Growth hormone releasing peptides (GHRPs) are synthetic peptides with the ability to stimulate human growth hormone (hGH) secretion. Several GHRPs have been developed as drug candidates; however, only one of them, GHRP-2 (Pralmorelin), has received a clinical approval.

source →
Laparoscopic Sleeve Gastrectomy Resolves Low GHRP-2-Stimulated Growth Hormone Levels in Obese Patients
Ohara E, Tokuyama H, Kitamoto T, Kitahara A, Hayashi A, Hayashi H, Takemoto M, Yokote K. · Obesity surgery (2017) ·

Because growth hormone (GH) secretion is reportedly decreased in obese patients, we examined not only the factors associated with the decreased GH secretion but also GH response to the GH-releasing peptide (GHRP)-2-load test before and after laparoscopic gastrectomy (LSG).

source →
Effects of GHRP-2 and Cysteamine Administration on Growth Performance, Somatotropic Axis Hormone and Muscle Protein Deposition in Yaks (Bos grunniens) with Growth Retardation
Hu R, Wang Z, Peng Q, Zou H, Wang H, Yu X, Jing X, Wang Y, Cao B, Bao S, Zhang W, Zhao S, Ji H, Kong X, Niu Q. · PloS one (2016) · rct

Unlabelled The objective of this study was to investigate the effects of growth hormone-releasing peptide-2 (GHRP-2) and cysteamine (CS) administration on growth performance in yaks with growth retardation and try to elucidate its regulatory mechanisms.

source →
Detection of GHRP-2 and GHRP-6 in urine samples from athletes
Cox HD, Hughes CM, Eichner D. · Drug testing and analysis (2015) ·
source →
Ghrelin receptor agonist, GHRP-2, produces antinociceptive effects at the supraspinal level via the opioid receptor in mice
Zeng P, Li S, Zheng YH, Liu FY, Wang JL, Zhang DL, Wei J. · Peptides (2014) · animal

GHRP-2 is a synthetic agonist of ghrelin receptor. GHRP-2 has similar physiological functions with ghrelin. In our previous study, ghrelin (i.c.v.) could induce analgesic effect through an interaction with GHS-R1α and with the central opioid system in the acute pain in mice.

source →